(19)
(11) EP 0 973 749 A1

(12)

(43) Date of publication:
26.01.2000 Bulletin 2000/04

(21) Application number: 98902513.5

(22) Date of filing: 13.01.1998
(51) International Patent Classification (IPC)7C07D 235/06, A61K 31/415, C07D 235/08, C07D 235/10, C07D 409/12, C07D 401/12, A61K 31/47
(86) International application number:
PCT/US9800/613
(87) International publication number:
WO 9835/945 (20.08.1998 Gazette 1998/33)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE
Designated Extension States:
AL LT LV RO SI

(30) Priority: 18.02.1997 US 801276

(71) Applicant: AMERICAN HOME PRODUCTS CORPORATION
Madison, New Jersey 07940-0874 (US)

(72) Inventors:
  • NELSON, James, Albert
    Washington Crossing, PA 18977 (US)
  • MEWSHAW, Richard, Eric
    Princeton, NJ 08540 (US)

(74) Representative: Mannion, Sally Kim, Dr. et al
c/o Wyeth Laboratories,Huntercombe Lane South,Taplow
Maidenhead,Berkshire SL6 0PH
Maidenhead,Berkshire SL6 0PH (GB)

   


(54) 4-AMINOALKOXY-1H-BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINE AUTORECEPTOR (D2) AGONISTS