(19)
(11) EP 1 000 055 A1

(12)

(43) Date of publication:
17.05.2000 Bulletin 2000/20

(21) Application number: 98923642.7

(22) Date of filing: 22.05.1998
(51) International Patent Classification (IPC)7C07D 401/04, A61K 31/415, A61K 31/44, A61K 31/505, C07D 401/14, C07D 409/14, C07D 413/14, C07D 405/14, C07D 471/04, C07D 417/14, C07D 453/02
(86) International application number:
PCT/US9810/436
(87) International publication number:
WO 9852/940 (26.11.1998 Gazette 1998/47)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 22.05.1997 US 47570 P

(71) Applicant: G.D. Searle & Co.
ChicagoIllinois 60680 (US)

(72) Inventors:
  • ANANTANARAYAN, Ashok
    Hainesville, IL 60030 (US)
  • CLARE, Michael
    Skokie, IL 60077 (US)
  • COLLINS, Paul, W.
    Deerfield, IL 60015 (US)
  • CRICH, Joyce, Zuowu
    Glenview, IL 60025 (US)
  • DEVRAJ, Rajesh
    Chesterfield, MO 63017 (US)
  • FLYNN, Daniel, L.
    Clarkson Valley, MO 63005 (US)
  • GENG, Lifeng
    Skokie, IL 60077 (US)
  • HANSON, Gunnar, J.
    Skokie, IL 60076 (US)
  • KOSZYK, Francis, J.
    Prospect Heights, IL 60070 (US)
  • LIAO, Shuyuan
    Glen Ellyn, IL 60137 (US)
  • PARTIS, Richard, A.
    Evanston, IL 60201 (US)
  • RAO, Shashidhar, N.
    Mundelein, IL 60060 (US)
  • SELNESS, Shaun, Raj
    St. Louis, MO 63141 (US)
  • SOUTH, Michael, S.
    St. Louis, MO 63146 (US)
  • STEALEY, Michael, A.
    Libertyville, IL 60048 (US)
  • WEIER, Richard, M.
    Lake Bluff, IL 60044 (US)
  • XU, Xiangdong
    Evanston, IL 60202 (US)
  • KHANNA, Ish K.
    Libertyville, IL 60048 (US)
  • YU, Yi
    Skokie, IL 60077 (US)

(74) Representative: Ebner von Eschenbach, Jennifer et al
c/o Ladas & Parry,Dachauerstrasse 37
80335 München
80335 München (DE)

   


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