(19)
(11) EP 1 001 969 A1

(12)

(43) Date of publication:
24.05.2000 Bulletin 2000/21

(21) Application number: 98939556.1

(22) Date of filing: 29.06.1998
(51) International Patent Classification (IPC)7C07K 5/00
(86) International application number:
PCT/EP9803/970
(87) International publication number:
WO 9901/470 (14.01.1999 Gazette 1999/02)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 30.06.1997 IT MI971545

(71) Applicants:
  • ZAMBON GROUP S.p.A.
    I-36100 Vicenza (IT)
  • INSTITUT NATIONAL DE LA SANTE ET DE LARECHERCHE MEDICALE (INSERM)
    75654 Paris CĂ©dex 13 (FR)

(72) Inventors:
  • UNGHERI, Domenico
    I-20015 Parabiago (IT)
  • PELLACINI, Franco
    I-20151 Milano (IT)
  • ROMAGNANO, Stefano
    I-20090 Buccinasco (IT)
  • KRAUS, Jean-Louis
    F-06540 Loda de Lantosque (FR)
  • CHERMANN, Jean-Claude
    F-13260 Cassis (FR)

(74) Representative: Longoni, Alessandra et al
c/o Zambon Group S.p.A.,Corp. Patent & Trademark Dept.,Via Lillo del Duca 10
20091 Bresso (Milano)
20091 Bresso (Milano) (IT)

   


(54) PEPTIDOMIMETIC DERIVATIVES SUICIDAL INHIBITORS OF THE HIV PROLIFERATION