(19)
(11) EP 1 012 150 A1

(12)

(43) Date of publication:
28.06.2000 Bulletin 2000/26

(21) Application number: 98924794.5

(22) Date of filing: 18.05.1998
(51) International Patent Classification (IPC)7C07D 413/02, C07D 231/12, C07D 261/18, C07D 261/08
(86) International application number:
PCT/US9810/174
(87) International publication number:
WO 9852/944 (26.11.1998 Gazette 1998/47)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 19.05.1997 US 47084 P
19.05.1997 US 46945 P
20.08.1997 US 56623 P
10.10.1997 US 61590 P

(71) Applicant: Sugen, Inc.
Redwood City, CA 94063 (US)

(72) Inventors:
  • McMAHON, Gerald
    Kenwood, CA 95452 (US)
  • TANG, Peng, Cho
    Moraga, CA 94556 (US)
  • SHAWVER, Laura, Kay
    San Francisco, CA 94112 (US)
  • HIRTH, Klaus, Peter
    San Francisco, CA 94114 (US)

(74) Representative: Viering, Jentschura & Partner 
Postfach 22 14 43
80504 München
80504 München (DE)

   


(54) HETEROARYLCARBOXAMIDE COMPOUNDS ACTIVE AGAINST PROTEIN TYROSINE KINASE RELATED DISORDERS