SYNTHESIS OF CLASTO-LACTACYSTIN BETA-LACTONE AND ANALOGS THEREOF - Patent 1021407

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EP 1 021 407 A1

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(43)	Date of publication:
	26.07.2000 Bulletin 2000/30

(21)	Application number: 98940885.1

(22)	Date of filing: 14.08.1998

(51)	International Patent Classification (IPC)⁷: C07D 207/46, C07D 263/14

(86)	International application number:
	PCT/US9816/858

(87)	International publication number:
	WO 9909/006 (25.02.1999 Gazette 1999/08)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

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Priority:

15.08.1997 US 55848 P
15.08.1997 US 912111
03.12.1997 US 67352 P

(71)	Applicant: Millennium Pharmaceuticals, Inc.
	Cambridge,Massachusetts 02139 (US)

(72)	Inventors:
	SOUCY, Francois Medford, MA 02155 (US) PLAMONDON, Louis Watertown, MA 02472-4922 (US) BEHNKE, Mark Somerville, MA 02144 (US) ROUSH, William Ann Arbor, MI 48105 (US)

(74)	Representative: Vossius, Volker, Dr. et al
	Dr. Volker Vossius,Patentanwaltskanzlei - Rechtsanwaltskanzlei,Holbeinstrasse 5 81679 München 81679 München (DE)

(54)	SYNTHESIS OF CLASTO-LACTACYSTIN BETA-LACTONE AND ANALOGS THEREOF