(19)
(11) EP 1 039 915 A1

(12)

(43) Date of publication:
04.10.2000 Bulletin 2000/40

(21) Application number: 98953531.5

(22) Date of filing: 14.10.1998
(51) International Patent Classification (IPC)7A61K 31/675, A61K 31/66, C07F 9/6574, C07F 9/6541, C07F 9/6533, C07F 9/653, C07F 9/59, C07F 9/58
(86) International application number:
PCT/US9821/750
(87) International publication number:
WO 9921/564 (06.05.1999 Gazette 1999/18)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 28.10.1997 US 63347 P

(71) Applicant: BRISTOL-MYERS SQUIBB COMPANY
Princeton, NJ 08543-4000 (US)

(72) Inventor:
  • SULSKY, Richard, B.
    West Trenton, NJ 08628 (US)

(74) Representative: VOSSIUS & PARTNER 
Siebertstrasse 4
81675 München
81675 München (DE)

   


(54) CYCLIC PHOSPHONATE ESTER INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND METHOD