QUINOLINEPIPERAZINE AND QUINOLINEPIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS COMBINED 5-HT1A, 5-HT1B AND 5-HT1D RECEPTOR ANTAGONISTS - Patent 1047691

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EP 1 047 691 A1

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(43)	Date of publication:
	02.11.2000 Bulletin 2000/44

(21)	Application number: 98965729.1

(22)	Date of filing: 02.12.1998

(51)	International Patent Classification (IPC)⁷: C07D 401/12, A61K 31/47, C07D 215/42, C07D 215/46, C07D 413/12, A61K 31/505, C07D 471/04 // (C07D471/04, 221:00), C07D209:00,(C07D471/04, 221:00), C07D221:00

(86)	International application number:
	PCT/EP9807/804

(87)	International publication number:
	WO 9931/086 (24.06.1999 Gazette 1999/25)

(84)	Designated Contracting States:
	BE CH DE ES FR GB IT LI NL

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Priority:

12.12.1997 GB 9726364
19.12.1997 GB 9726905
07.01.1998 GB 9800317

(71)	Applicant: SMITHKLINE BEECHAM PLC
	Brentford,Middlesex TW8 9EP (GB)

(72)	Inventor:
	GASTER, Laramie, Mary,SmithKline Beecham Pharm. Harlow,Essex CM19 5AW (GB)

(74)	Representative: Waters, David Martin, Dr. et al
	Smithkline Beecham plcCorporate Intellectual Property,Two New Horizons Court Brentford, Middlesex TW8 9EP Brentford, Middlesex TW8 9EP (GB)

(54)	QUINOLINEPIPERAZINE AND QUINOLINEPIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS COMBINED 5-HT1A, 5-HT1B AND 5-HT1D RECEPTOR ANTAGONISTS