(19)
(11) EP 1 054 876 A1

(12)

(43) Date of publication:
29.11.2000 Bulletin 2000/48

(21) Application number: 98958896.7

(22) Date of filing: 27.10.1998
(51) International Patent Classification (IPC)7: C07D 285/12, A61K 31/41, C07D 401/12, A61K 31/44, C07D 403/12, C07D 403/04, A61K 31/55
(86) International application number:
PCT/EP9806/995
(87) International publication number:
WO 9928/309 (10.06.1999 Gazette 1999/23)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 26.11.1997 GB 9725055

(71) Applicant: PHARMACIA & UPJOHN S.p.A.
20152 Milano (IT)

(72) Inventors:
  • PEVARELLO, Paolo
    I-27100 Pavia (IT)
  • AMICI, Raffaella
    I-20073 Codogno (IT)
  • VILLA, Manuela
    I-22040 Lurago d'Erba (IT)
  • TOMA, Salvatore
    I-20146 Milano (IT)
  • VARASI, Mario
    I-20100 Milano (IT)

   


(54) 1,3,4-THIADIAZOLES DERIVATIVES AS KYN-OH INHIBITORS