META-AZACYCLIC AMINO BENZOIC ACID COMPOUNDS AND DERIVATIVES THEREOF BEING INTEGRIN ANTAGONISTS - Patent 1060164

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EP 1 060 164 A1

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(43)	Date of publication:
	20.12.2000 Bulletin 2000/51

(21)	Application number: 99937927.4

(22)	Date of filing: 22.02.1999

(51)	International Patent Classification (IPC)⁷: C07D 233/26, A61K 31/505

(86)	International application number:
	PCT/US9903/281

(87)	International publication number:
	WO 9944/994 (10.09.1999 Gazette 1999/36)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

04.03.1998 US 34270

(71)	Applicant: G.D. SEARLE & CO.
	Chicago, IL 60680-5110 (US)

(72)	Inventors:
	ROGERS, Thomas, E. Ballwin, MO 63021 (US) RUMINSKI, Peter, G. Dardeene Prairie, MO 63366 (US)

(74)	Representative: Ebner von Eschenbach, Jennifer et al
	c/o Ladas & Parry,Dachauerstrasse 37 80335 München 80335 München (DE)

(54)	META-AZACYCLIC AMINO BENZOIC ACID COMPOUNDS AND DERIVATIVES THEREOF BEING INTEGRIN ANTAGONISTS