(19)
(11) EP 1 062 199 A1

(12)

(43) Date of publication:
27.12.2000 Bulletin 2000/52

(21) Application number: 99907333.1

(22) Date of filing: 11.03.1999
(51) International Patent Classification (IPC)7C07C 235/84, C07D 213/55, C07D 239/28, C07D 241/24, A61K 31/17, A61K 31/44, A61K 31/50, A61K 31/505
(86) International application number:
PCT/DK9900/122
(87) International publication number:
WO 9946/236 (16.09.1999 Gazette 1999/37)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE

(30) Priority: 12.03.1998 DK 34298
12.03.1998 DK 34598
03.04.1998 DK 47298
03.04.1998 DK 47998
15.07.1998 DK 94098

(71) Applicants:
  • NOVO NORDISK A/S
    2880 Bagsvaerd (DK)
  • Ontogen Corporation
    Carlsbad, CA 92009 (US)

(72) Inventors:
  • RICHTER, Lutz Stefan
     (DK)
  • ANDERSEN, Henrik, Sune
    DK-2800 Lyngby (DK)
  • VAGNER, Josef
    DK-3500 Vaerloese (DK)
  • JEPPESEN, Claus, Bekker
    DK-2990 Nivaa (DK)
  • MOLLER, Niels, Peter, Hundahl
    DK-2100 Copenhagen (DK)
  • BRANNER, Sven
    DK-2800 Lyngby (DK)
  • SU, Jing
    New York, NY 10021 (US)
  • BAKIR, Farid
    San Diego, CA 92120 (US)
  • JUDGE, Luke, Milburn
    La Jolla, CA 92037 (US)

   


(54) MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES)