(19)
(11) EP 1 062 222 A1

(12)

(43) Date of publication:
27.12.2000 Bulletin 2000/52

(21) Application number: 99911781.5

(22) Date of filing: 09.03.1999
(51) International Patent Classification (IPC)7C07F 9/572, A61K 31/675, G01N 33/58, C07F 9/40, C07F 9/6571
(86) International application number:
PCT/EP9901/617
(87) International publication number:
WO 9946/272 (16.09.1999 Gazette 1999/37)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE
Designated Extension States:
LT LV SI

(30) Priority: 09.03.1998 EP 98200733

(71) Applicant: Fondatech Benelux N.V.
2140 Borgerhout (BE)

(72) Inventors:
  • SCHARPE, Simon, Lodewijk
    B-2610 Antwerpen (BE)
  • DE MEESTER, Ingrid, Anna, Jozef
    B-2610 Wilrijk (BE)
  • BELIAEV, Alexandre Arkadicvitch;
    P-4480 Mindelo-Vila-Do Conde (PT)
  • LAMBEIR, Anne-Marie, Virginie, RenĂ©e
    B-3001 Heverlee (BE)
  • AUGUSTYNS, Koen, Jan, Ludovicus
    B-2322 Minderhout (BE)
  • HAEMERS, Achiel, Jean-Marie
    B-9830 Sint-Martens-Latem (BE)
  • GOOSSENS, Filip, Jozef, Anny
    B-1910 Kampenhout (BE)
  • HENDRIKS, Dirk, Frans
    B-2360 Aartselaar (BE)

(74) Representative: Van Someren, Petronella F. H. M. et al
Arnold & Siedsma,Advocaten en Octrooigemachtigden,Sweelinckplein 1
2517 GK Den Haag
2517 GK Den Haag (NL)

   


(54) SERINE PEPTIDASE MODULATORS