(19)
(11) EP 1 066 039 A1

(12)

(43) Date of publication:
10.01.2001 Bulletin 2001/02

(21) Application number: 99911063.8

(22) Date of filing: 02.03.1999
(51) International Patent Classification (IPC)7A61K 31/50, A61K 31/505, C07D 237/26, C07D 239/70, C07D 491/04, C07D 491/048, C07D 491/056, C07D 498/04
(86) International application number:
PCT/US9904/609
(87) International publication number:
WO 9944/612 (10.09.1999 Gazette 1999/36)
(84) Designated Contracting States:
BE CH DE ES FR GB IE IT LI NL

(30) Priority: 02.03.1998 US 76451 P

(71) Applicant: CoCensys, Inc.
Irvine, CA 92618 (US)

(72) Inventors:
  • UPASANI, Ravi
    Foothill Ranch, CA 92610 (US)
  • CAI, Sui, X.
    San Diego, CA 92121 (US)
  • LAN, Nancy, C.
    S. Pasadena, CA 91030 (US)
  • WANG, Yan
    San Diego, CA 92129 (US)
  • FIELD, George
    Danville, CA 94526 (US)
  • FICK, David, B.
    Mission Viejo, CA 92691 (US)

(74) Representative: Chapman, Paul William et al
Kilburn & Strode,20 Red Lion Street
London WC1R 4PJ
London WC1R 4PJ (GB)

   


(54) SUBSTITUTED QUINAZOLINES AND ANALOGS AND THE USE THEREOF