(19)
(11) EP 1 068 207 A1

(12)

(43) Date of publication:
17.01.2001 Bulletin 2001/03

(21) Application number: 99916294.4

(22) Date of filing: 01.04.1999
(51) International Patent Classification (IPC)7C07D 471/04, C07D 487/04, A61K 31/435, A61K 31/505
// (C07D487/04, 239:00), C07D209:00,(C07D471/04, 221:00), C07D209:00
(86) International application number:
PCT/US9907/254
(87) International publication number:
WO 9951/600 (14.10.1999 Gazette 1999/41)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 02.04.1998 US 80451 P

(71) Applicant: NEUROGEN CORPORATION
Branford, CT 06405 (US)

(72) Inventors:
  • HORVATH, Raymond, F.
    North Branford, CT 06471 (US)
  • DARROW, James, W.
    Wallingford, CT 06492 (US)
  • MAYNARD, George, D.
    Clinton, CT 06413 (US)

(74) Representative: Eyles, Christopher Thomas 
W.P. THOMPSON & CO.Celcon House289-293 High Holborn
London WC1V 7HU
London WC1V 7HU (GB)

   


(54) AMINOALKYL SUBSTITUTED 9H-PYRIDINO 2,3-b]INDOLE AND 9H-PYRIMIDINO 4,5-b]INDOLE DERIVATIVES