(19)
(11) EP 1 070 060 A1

(12)

(43) Date of publication:
24.01.2001 Bulletin 2001/04

(21) Application number: 99916119.3

(22) Date of filing: 09.04.1999
(51) International Patent Classification (IPC)7: C07D 401/12, A61K 31/44, C07K 5/023, C07D 213/82, C07D 495/10, C07D 409/12, C07D 333/38, C07D 403/12, C07D 417/12
(86) International application number:
PCT/US9904/297
(87) International publication number:
WO 9952/896 (21.10.1999 Gazette 1999/42)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

(30) Priority: 10.04.1998 US 81394 P

(71) Applicant: G.D. Searle & Co.
Chicago, IL 60606-5110 (US)

(72) Inventors:
  • CHANDRAKUMAR, Nizal, Samuel
    Vernon Hills, IL 60061 (US)
  • DESAI, Bipinchandra, Nanubhai
    Vernon Hills, IL 60061 (US)
  • DEVADAS, Balekudru
    Chesterfield, MO 63017 (US)
  • HUFF, Renee
    Park Ridge, IL 60068 (US)
  • KHANNA, Ish, K.
    Vernon Hills, IL 60061 (US)
  • RAO, Shashidhar, N.
    Mundelein, IL 60060 (US)
  • RICO, Joseph, G.
    Ballwin, MO 63021 (US)
  • ROGERS, Thomas, E.
    Ballwin, MO 63021 (US)
  • RUMINSKI, Peter, G.
    Dardenne Prairie, MO 63366 (US)
  • RUSSELL, Mark, Andrew
    Gurnee, IL 60031 (US)
  • YU, Yi
    Skokie, IL 60077 (US)
  • GASIECKI, Alan, Frank
    Vernon Hills, IL 60061 (US)
  • MALECHA, James, W.
    Libertyville, IL 60048 (US)
  • MIYASHIRO, Julie, M.
    Skokie, IL 60076 (US)

(74) Representative: Albrecht, Thomas, Dr. et al
Kraus & Weisert,Thomas-Wimmer-Ring 15
80539 München
80539 München (DE)

   


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