(19)
(11) EP 1 080 068 A1

(12)

(43) Date of publication:
07.03.2001 Bulletin 2001/10

(21) Application number: 99907336.4

(22) Date of filing: 12.03.1999
(51) International Patent Classification (IPC)7C07C 235/84
(86) International application number:
PCT/DK9900/126
(87) International publication number:
WO 9946/237 (16.09.1999 Gazette 1999/37)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE
Designated Extension States:
LT RO SI

(30) Priority: 12.03.1998 DK 35098
12.03.1998 DK 34598
12.03.1998 DK 34398
12.03.1998 DK 34298
12.03.1998 DK 34498
12.03.1998 DK 34798
12.03.1998 DK 34698
12.03.1998 DK 34898
03.04.1998 DK 47998
03.04.1998 DK 47298
03.04.1998 DK 47398
03.04.1998 DK 47898
03.04.1998 DK 47598
03.04.1998 DK 47498
03.04.1998 DK 47698
03.04.1998 DK 48098
24.04.1998 US 82912 P
15.05.1998 DK 66798
05.06.1998 US 88115 P
15.07.1998 DK 93998
15.07.1998 DK 94098
15.07.1998 DK 93898
28.10.1998 DK 138598
26.11.1998 DK 156198
07.12.1998 DK 161298

(71) Applicants:
  • Novo Nordisk A/S
    2880 Bagsvaerd (DK)
  • Ontogen Corporation
    Carlsbad, CA 92009 (US)

(72) Inventors:
  • RICHTER, Lutz Stefan
    DECEASED (DK)
  • ANDERSEN, Henrik Sune
    2800 Lyngby (DK)
  • VAGNER, Josef
    Oro Valley, AZ 85737 (US)
  • JEPPESEN, Claus, Becker
    2900 Nivaamolen (DK)
  • MOELLER, Niels P H
    2100 Copenhagen (DK)
  • BRANNER, Sven
    2800 Lyngby (DK)
  • JEPPESEN, Lone
    2830 Virum (DK)
  • OLSEN, Ole Hvilsted
    2700 Broenshoej (DK)
  • IVERSEN, Lars Fogh
    2840 Holte (DK)
  • HOLSWORTH, Daniel Dale
    San Diego, CA 92129 (US)
  • AXE, Frank Urban
    Escondido, CA 92027 (US)
  • GE, Yu
    San Diego, CA 92129 (US)
  • JONES, Todd, Kevin
    Solana Beach, CA 92075 (US)
  • RIPKA, William Charles
    San Diego, CA 92131 (US)
  • UYEDA, Roy Teruyuki
    San Diego, CA 92122 (US)
  • SU, Jing
    New York, NY 10021 (US)
  • BAKIR, Farid
    San Diego, CA 92120 (US)
  • JUDGE, Luke Milburn
    La Jolla, CA 92037 (US)

(74) Representative: Stephensen, Birgitte Borregaard (DK) 
c/o Novo Nordisk A/SCorporate PatentsNovo Allé
2880 Bagsvaerd
2880 Bagsvaerd (DK)

   


(54) MODULATORS OF PROTEIN TYROSINE PHOSPHATASES