(19)
(11) EP 1 084 149 A1

(12)

(43) Date of publication:
21.03.2001 Bulletin 2001/12

(21) Application number: 99922527.9

(22) Date of filing: 27.05.1999
(51) International Patent Classification (IPC)7C08B 37/16, A61K 47/48
(86) International application number:
PCT/JP9902/806
(87) International publication number:
WO 9962/958 (09.12.1999 Gazette 1999/49)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE
Designated Extension States:
LT LV MK RO SI

(30) Priority: 29.05.1998 JP 16446598

(71) Applicant: JANSSEN PHARMACEUTICA N.V.
2340 Beerse (BE)

(72) Inventors:
  • UEKAMA, Kaneto
    Kumamoto-shi,Kumamoto 862-0938 (JP)
  • HIRAYAMA, Fumitoshi
    Kumamoto-shi,Kumamoto 862-0909 (JP)
  • KONDO, Akira
    Sunto-gun,Shizuoka 411-0932 (JP)
  • KAWAJI, Hiroshi
    Sunto-gun,Shizuoka 411-0932 (JP)
  • OHTA, Masaaki
    Sunto-gun,Shizuoka 411-0932 (JP)
  • OKAMOTO, Yasuhiro
    Sunto-gun,Shizuoka 411-0932 (JP)

(74) Representative: Quaghebeur, Luc et al
Janssen Pharmaceutica N.V.,Patent Department,Turnhoutseweg 30
2340 Beerse
2340 Beerse (BE)

   


(54) ACYLATED ALKYLATED CYCLODEXTRIN DERIVATIVES AND THEIR USE AS CARRIERS FOR MEDICAMENTS