MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5-HT 3? RECEPTORS - Patent 1085888

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EP 1 085 888 A1

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(43)	Date of publication:
	28.03.2001 Bulletin 2001/13

(21)	Application number: 99928450.8

(22)	Date of filing: 08.06.1999

(51)	International Patent Classification (IPC)⁷: A61K 38/00, A61K 39/00, A61K 39/44, A61K 39/395, A61K 51/00, C07K 2/00, C07K 4/00, G01N 33/53, G01N 33/543, G01N 33/566

(86)	International application number:
	PCT/US9912/768

(87)	International publication number:
	WO 9964/046 (16.12.1999 Gazette 1999/50)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

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Priority:

08.06.1998 US 88466 P
15.07.1998 US 92938 P
16.02.1999 US 120282 P

(71)	Applicant: Advanced Medicine, Inc.
	South San Francisco, CA 94080 (US)

(72)	Inventors:
	YANG, Guang San Mateo, CA 94402 (US) MEIER-DAVIS, Susan Belmont, CA 94002 (US) GRIFFIN, John, H. Atherton, CA 94027 (US)

(74)	Representative: Hay, Martin Alexander et al
	Martin A. Hay & Co.13 Queen Victoria Street MacclesfieldCheshire SK11 6LP MacclesfieldCheshire SK11 6LP (GB)

(54)	MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5-HT 3? RECEPTORS