(19)
(11) EP 1 094 814 A2

(12)

(88) Date of publication A3:
03.02.2000

(43) Date of publication:
02.05.2001 Bulletin 2001/18

(21) Application number: 99927848.4

(22) Date of filing: 03.06.1999
(51) International Patent Classification (IPC)7A61K 31/47, A61K 31/34, A61K 31/495, A61K 31/425
(86) International application number:
PCT/EP9903/827
(87) International publication number:
WO 9964/001 (16.12.1999 Gazette 1999/50)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 05.06.1998 GB 9812189

(71) Applicant: GLAXO GROUP LIMITED
Greenford, Middlesex UB6 ONN (GB)

(72) Inventors:
  • BROUWER, Kenneth Russell
    Research Triangle Park, NC 27709 (US)
  • POLLI, Joseph, William
    Research Triangle Park, NC 27709 (US)

(74) Representative: Crawley, Karen Anne 
Glaxo Wellcome plc,Glaxo Wellcome House,Berkeley Avenue
Greenford,Middlesex UB6 0NN
Greenford,Middlesex UB6 0NN (GB)

   


(54) METHODS AND COMPOSITIONS FOR INCREASING PENETRATION OF HIV PROTEASE INHIBITORS