(19)
(11) EP 1 098 892 A1

(12)

(43) Date of publication:
16.05.2001 Bulletin 2001/20

(21) Application number: 99934632.3

(22) Date of filing: 08.07.1999
(51) International Patent Classification (IPC)7C07D 295/135, A61K 31/496, C07D 295/18, C07D 271/10, C07D 271/06, A61K 31/4245
(86) International application number:
PCT/EP9904/803
(87) International publication number:
WO 0005/225 (03.02.2000 Gazette 2000/05)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 20.07.1998 EP 98113488

(71) Applicant: MERCK PATENT GmbH
64293 Darmstadt (DE)

(72) Inventors:
  • BÖTTCHER, Henning
    D-64287 Darmstadt (DE)
  • VAN AMSTERDAM, Christoph
    D-64295 Darmstadt (DE)
  • HARTING, Jürgen
    D-64287 Darmstadt (DE)
  • WIKSTRÖM, Hakan, Vilhelm
    NL-9721 WN Groningen (NL)
  • LIAO, Yi
    NL-9742 GL Groningen (NL)

   


(54) BIPHENYL DERIVATIVES