(19)
(11) EP 1 104 413 A2

(12)

(88) Date of publication A3:
03.08.2000

(43) Date of publication:
06.06.2001 Bulletin 2001/23

(21) Application number: 99936874.9

(22) Date of filing: 04.08.1999
(51) International Patent Classification (IPC)7C07D 295/15, A61K 31/495, C07D 295/185, C07D 211/70
(86) International application number:
PCT/GB9902/560
(87) International publication number:
WO 0008/006 (17.02.2000 Gazette 2000/07)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 07.08.1998 GB 9817197

(71) Applicants:
  • ELI LILLY AND COMPANY LIMITED
    Basingstoke,Hants RG21 6XA (GB)
  • ELI LILLY AND COMPANY
    Indianapolis, Indiana 46285 (US)

(72) Inventors:
  • BAKER, Stephen Richard
    Yateley,Hampshire GU46 7DQ (GB)
  • BLEAKMAN, David
    Zionsville, IN 46077 (US)
  • GOLDSWORTHY, John
    Basingstoke,Hapshire RG24 9JW (GB)
  • HAHN, Patric, James
    Indianapolis, IN 46237 (US)
  • JAGDMANN, Gunnar, Erik
    Apex, NC 27502 (US)
  • TURKINGTON, Shelley, Hunnings
    Durham, NC 27705 (US)

(74) Representative: Denholm, Anna Marie et al
Eli Lilly and Company Limited,Lilli Research Centre,Erl Wood Manor
WindleshamSurrey GU20 6PH
WindleshamSurrey GU20 6PH (GB)

   


(54) PIPERIDINE AND PIPERAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUNDS CONTAINING THEM