(19)
(11) EP 1 124 802 A1

(12)

(43) Date of publication:
22.08.2001 Bulletin 2001/34

(21) Application number: 99951035.7

(22) Date of filing: 01.11.1999
(51) International Patent Classification (IPC)7C07D 211/76, C07D 211/22
(86) International application number:
PCT/IB9901/762
(87) International publication number:
WO 0026/187 (11.05.2000 Gazette 2000/19)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 02.11.1998 US 106673 P

(71) Applicant: Synthon B.V.
6545 CM Nijmegen (NL)

(72) Inventors:
  • PETERS, Theodorus, Hendricus, Antonius
    NL-6814 JB Arnhem (NL)
  • BENNEKER, Franciscus, Bernardus, Gemma
    NL-6991 HA Rheden (NL)
  • HOORN, Hans, Jan
    NL-6546 VX Nijmegen (NL)
  • PICHA, Frantisek
    615 00 Brno (CZ)

(74) Representative: Duxbury, Stephen 
Arnold & Siedsma,Sweelinckplein 1
2517 GK Den Haag
2517 GK Den Haag (NL)

   


(54) PROCESS FOR PRODUCING 4-ARYLPIPERIDINE-3-CARBINOLS AND RELATED COMPOUNDS