(19)
(11) EP 1 139 754 A1

(12)

(43) Date of publication:
10.10.2001 Bulletin 2001/41

(21) Application number: 99966725.6

(22) Date of filing: 30.12.1999
(51) International Patent Classification (IPC)7A01N 43/38, A61K 31/40
(86) International application number:
PCT/US9931/232
(87) International publication number:
WO 0038/519 (06.07.2000 Gazette 2000/27)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 31.12.1998 US 114313 P

(71) Applicant: Sugen, Inc.
South San Francisco, CA 94080-4811 (US)

(72) Inventors:
  • LANGECKER, Peter, J.
    Monte Sereno, CA 95030 (US)
  • SHAWVER, Laura, Kay
    San Francisco, CA 94112 (US)
  • TANG, Peng, Cho
    Moraga, CA 94556 (US)
  • SUN, Li
    Foster City, CA 94404 (US)

(74) Representative: Viering, Jentschura & Partner 
Postfach 22 14 43
80504 München
80504 München (DE)

   


(54) 3-HETEROARYLIDENYL-2-INDOLINONE COMPOUNDS FOR MODULATING PROTEIN KINASE ACTIVITY AND FOR USE IN CANCER CHEMOTHERAPY