(19)
(11) EP 1 140 902 A1

(12)

(43) Date of publication:
10.10.2001 Bulletin 2001/41

(21) Application number: 99963980.0

(22) Date of filing: 16.12.1999
(51) International Patent Classification (IPC)7C07D 401/14, C07D 413/14, C07D 407/14, A61K 31/445, A61K 31/44, A61K 31/55, A61P 35/00
(86) International application number:
PCT/US9927/939
(87) International publication number:
WO 0037/459 (29.06.2000 Gazette 2000/26)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 18.12.1998 US 216398

(71) Applicant: SCHERING CORPORATION
Kenilworth,New Jersey 07033-0530 (US)

(72) Inventors:
  • TAVERAS, Arthur, G.
    Denville, NJ 07834 (US)
  • DOLL, Ronald, J.
    Maplewood, NJ 07040 (US)
  • COOPER, Alan, B.
    West Caldwell, NJ 07006 (US)
  • FERREIRA, Johan, A.
    Bensalem, PA 19020 (US)
  • GUZI, Timothy
    Chatham, NJ 07928 (US)
  • MALLAMS, Alan, K.
    Hackettstown, NJ 07840-9302 (US)
  • RANE, Dinanath, F.
    Morganville, NJ 07751 (US)
  • GIRIJAVALLABHAN, Viyyoor, M.
    Parsippany, NJ 07054 (US)
  • AFONSO, Adriano
    West Caldwell, NJ 07006 (US)
  • AKI, Cynthia, J.
    Rutherford, NJ 07070 (US)
  • CHAO, Jianping
    Summit, NJ 07901 (US)
  • ALVAREZ, Carmen
    Roselle Park, NJ 07204 (US)
  • KELLY, Joseph, M.
    Parlin, NJ 08859 (US)
  • LALWANI, Tarik
    Philadelphia, PA 19107 (US)
  • DESAI, Jagdish, A.
    Spotswood, NJ 08884 (US)
  • WANG, James, J., S.
    Westfield, NJ 07090 (US)
  • WEINSTEIN, Jay
    Upper Montclair, NJ 07043 (US)

(74) Representative: Ritter, Stephen David et al
Mathys & Squire100 Gray's Inn Road
London WC1X 8AL
London WC1X 8AL (GB)

   


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