(19)
(11) EP 1 144 396 A2

(12)

(88) Date of publication A3:
09.11.2000

(43) Date of publication:
17.10.2001 Bulletin 2001/42

(21) Application number: 99968883.1

(22) Date of filing: 14.12.1999
(51) International Patent Classification (IPC)7: C07D 277/18, C07D 277/54, C07D 277/60, C07D 263/28, C07D 263/52, C07D 279/06, C07D 281/02, C07D 417/12, A61K 31/421, A61K 31/423, A61K 31/426, A61K 31/428, A61K 31/54, A61K 31/55
(86) International application number:
PCT/US9929/601
(87) International publication number:
WO 0042/031 (20.07.2000 Gazette 2000/29)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
LT LV RO SI

(30) Priority: 14.01.1999 US 231906

(71) Applicant: Bayer Corporation
Pittsburgh, PA 15205 (US)

(72) Inventors:
  • DIXON, Brian R.
    Woodbridge, CT 06525 (US)
  • BAGI, Cedo M.
    Branford, CT 06405 (US)
  • BRENNEN, Catherine R.
    Milford, CT 06460 (US)
  • BRITTELLI, David R.
    Branford, CT 06405 (US)
  • BULLOCK, William H.
    Easton, CT 06612 (US)
  • CHEN, Jinshan
    Hamden, Ct 06514 (US)
  • COLLIBEE, William L.
    Bethany, CT 06524 (US)
  • DALLY, Robert
    East Haven, CT 06513 (US)
  • JOHNSON, Jeffrey S.
    Branford, CT 06405 (US)
  • KLUENDER, Harold C. E.
    Trumbull, CT 06611 (US)
  • LATHROP, William F.
    Plantsville, CT 06479 (US)
  • LIU, Peiying
    Madison, CT 06443 (US)
  • MASE, Carol Ann
    Ringoes, NJ 08551 (US)
  • REDMAN, Aniko M.
    Derby, CT 06418 (US)
  • SCOTT, William J.
    Guilford, CT 06437 (US)
  • URBAHNS, Klaus
    D-42329 Wuppertal (DE)
  • WOLANIN, Donald J.
    Orange, CT 06477 (US)

(74) Representative: Welch, Andreas, Dr. et al
Bayer AG,Konzernbereich RP/PL
51368 Leverkusen
51368 Leverkusen (DE)

   


(54) SUBSTITUTED 2-ARYLIMINO HETEROCYCLES AND COMPOSITIONS CONTAINING THEM, FOR USE AS PROGESTERONE RECEPTOR BINDING AGENTS