(19)
(11) EP 1 144 404 A1

(12)

(43) Date of publication:
17.10.2001 Bulletin 2001/42

(21) Application number: 00902605.5

(22) Date of filing: 17.01.2000
(51) International Patent Classification (IPC)7C07D 401/06, C07D 401/12, C07D 401/14, A61K 31/445, A61K 31/47, A61P 31/04
(86) International application number:
PCT/EP0000/350
(87) International publication number:
WO 0043/383 (27.07.2000 Gazette 2000/30)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 20.01.1999 GB 9901236
08.10.1999 GB 9923936

(71) Applicant: SMITHKLINE BEECHAM PLC
Brentford,Middlesex TW8 9EP (GB)

(72) Inventors:
  • DAVIES, David, Thomas,SmithKline Beecham Pharm.
    Harlow,Essex CM19 5AW (GB)
  • HENRY, Caroline, Joan,SmitKline Beecham Pharm.
    Harlow,Essex CM19 5AW (GB)
  • PEARSON, Neil, David,SmithKline Beecham Pharm.
    Harlow,Essex CM19 5AW (GB)

(74) Representative: Valentine, Jill Barbara et al
GlaxoSmithKline,Two New Horizons Court
Brentford, Middlesex TW8 9EP
Brentford, Middlesex TW8 9EP (GB)

   


(54) PIPERIDINYLQUINOLINES AS PROTEIN TYROSINE KINASE INHIBITORS