CRYSTALLINE FORM OF BENZOQUINOLINE-3-ONE DERIVATIVE AS INHIBITOR OF 5-ALPHA REDUCTASE - Patent 1149080

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EP 1 149 080 A2

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(88)	Date of publication A3:
	18.01.2001

(43)	Date of publication:
	31.10.2001 Bulletin 2001/44

(21)	Application number: 99964980.9

(22)	Date of filing: 10.11.1999

(51)	International Patent Classification (IPC)⁷: C07D 221/00, A61K 31/473, A61P 35/00

(86)	International application number:
	PCT/US9926/809

(87)	International publication number:
	WO 0034/245 (15.06.2000 Gazette 2000/24)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

07.12.1998 US 111243 P

(71)	Applicant: ELI LILLY AND COMPANY
	Indianapolis, Indiana 46285 (US)

(72)	Inventor:
	WEIGEL, Leland, Otto Indianapolis, IN 46254 (US)

(74)	Representative: Burnside, Ivan John et al
	Eli Lilly and Company LimitedLilly Research CentreErl Wood Manor Windlesham, Surrey GU20 6PH Windlesham, Surrey GU20 6PH (GB)

(54)	CRYSTALLINE FORM OF BENZOQUINOLINE-3-ONE DERIVATIVE AS INHIBITOR OF 5-ALPHA REDUCTASE