(19)
(11) EP 1 150 955 A2

(12)

(88) Date of publication A3:
01.03.2001

(43) Date of publication:
07.11.2001 Bulletin 2001/45

(21) Application number: 00907184.6

(22) Date of filing: 03.02.2000
(51) International Patent Classification (IPC)7: C07D 213/75, C07D 213/65, C07D 405/14, C07D 409/14, C07D 213/81, C07D 213/82, C07C 233/75, A61K 31/4427, A61K 31/16, A61P 25/00, A61P 29/00
(86) International application number:
PCT/US0003/042
(87) International publication number:
WO 0046/203 (10.08.2000 Gazette 2000/32)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 04.02.1999 US 118893 P

(71) Applicant: Millennium Pharmaceuticals, Inc.
Cambridge,Massachusetts 02139 (US)

(72) Inventors:
  • SHIOSAKI, Kazumi
    Wellesley, MA 02481 (US)
  • FLEMING, Paul
    Somerville, MA 02143 (US)

(74) Representative: Plougmann, Vingtoft & Partners 
Sankt Annae Plads 11
1250 Copenhagen K
1250 Copenhagen K (DK)

   


(54) G-PROTEIN COUPLED HEPTAHELICAL RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF