(19)
(11)
EP 1 155 001 A1
(12)
(43)
Date of publication:
21.11.2001
Bulletin 2001/47
(21)
Application number:
00919327.7
(22)
Date of filing:
18.02.2000
(51)
International Patent Classification (IPC)
7
:
C07D
217/02
,
C07D
217/24
,
A61K
31/47
(86)
International application number:
PCT/US0004/316
(87)
International publication number:
WO 0050/406
(
31.08.2000
Gazette 2000/35)
(84)
Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
(30)
Priority:
22.02.1999
US 255396
17.02.2000
US 506853
(71)
Applicant:
TREGA BIOSCIENCES, INC.
San Diego, CA 92121 (US)
(72)
Inventor:
LEBL, Michael
San Diego, CA 92121 (US)
(74)
Representative:
Schohe, Stefan
Forrester & BoehmertPettenkoferstrasse 20-22
80336 München
80336 München (DE)
(54)
ISOQUINOLINE DERIVATIVES AND ISOQUINOLINE COMBINATORIAL LIBRARIES