(19)

(11)

EP 1 155 021 A1

(12)

(43) Date of publication: 21.11.2001 Bulletin 2001/47 (21) Application number: 00904573.3 (22) Date of filing: 26.01.2000

(51) International Patent Classification (IPC)7: C07F 9/06, C07D 311/04, A61K 9/00, A61K 31/66, A61K 31/35 (86) International application number: PCT/US0001/923 (87) International publication number: WO 0044/757 (03.08.2000 Gazette 2000/31)

(84) Designated Contracting States: AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE Designated Extension States: AL LT LV MK RO SI (30) Priority: 27.01.1999 US 117567 P 01.02.1999 US 118198 P (71) Applicant: Zielinski Laboratory San Diego, CA 92121 (US)	(72) Inventor: ZIELINSKI, Jan, E. Vista, CA 92083 (US) (74) Representative: VOSSIUS & PARTNER  Siebertstrasse 4 81675 München 81675 München (DE)