ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS - Patent 1157003

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EP 1 157 003 A1

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(43)	Date of publication:
	28.11.2001 Bulletin 2001/48

(21)	Application number: 00903853.0

(22)	Date of filing: 16.02.2000

(51)	International Patent Classification (IPC)⁷: C07C 255/29, C07C 255/25, C07D 307/54, C07D 231/12, C07D 295/08, C07C 323/60, A61K 31/275, A61K 31/33, A61P 19/00, C07D 333/24, C07D 249/18

(86)	International application number:
	PCT/GB0000/539

(87)	International publication number:
	WO 0048/992 (24.08.2000 Gazette 2000/34)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

20.02.1999 GB 9903861

(71)	Applicant: AstraZeneca AB
	151 85 Södertälje (SE)

(72)	Inventors:
	TUCKER, Howard Macclesfield,Cheshire SK10 4TG (GB) LARGE, Michael Stewart Macclesfield,Cheshire SK10 4TG (GB) OLDFIELD, John Macclesfield,Cheshire SK10 4TG (GB) JOHNSTONE, Craig Macclesfield,Cheshire SK10 4TG (GB) EDWARDS, Philip Neil Macclesfield,Cheshire SK10 4TG (GB)

(74)	Representative: Tierney, Francis John et al
	AstraZeneca UK Limited,Global Intellectual Property Patents,P.O. Box 272,Mereside,Alderley Park Macclesfield,Cheshire SK10 4GR Macclesfield,Cheshire SK10 4GR (GB)

(54)	ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS