(19)
(11) EP 1 159 268 A1

(12)

(43) Date of publication:
05.12.2001 Bulletin 2001/49

(21) Application number: 00917652.0

(22) Date of filing: 22.02.2000
(51) International Patent Classification (IPC)7C07D 209/12, A61K 31/40, A61P 19/10
(86) International application number:
PCT/US0004/386
(87) International publication number:
WO 0051/983 (08.09.2000 Gazette 2000/36)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 04.03.1999 US 262413

(71) Applicant: AMERICAN HOME PRODUCTS CORPORATION
Madison, New Jersey 07940-0874 (US)

(72) Inventors:
  • KOKO, Marci, Catherine
    Wayne, PA 19087 (US)
  • ULLRICH, John, William
    Schwenksville, PA 19473 (US)
  • SANTILLI, Arthur, Attilio
    Havertown, PA 19083 (US)

(74) Representative: Wileman, David Francis Dr. et al
c/o Patent DepartmentWyeth LaboratoriesHuntercombe Lane South
TaplowMaidenheadBerkshire SL6 OPH
TaplowMaidenheadBerkshire SL6 OPH (GB)

   


(54) N-SUBSTITUTED BENzOYL INDOLES AS ESTROGENIC AGENTS