(19)
(11) EP 1 165 076 A1

(12)

(43) Date of publication:
02.01.2002 Bulletin 2002/01

(21) Application number: 00912193.0

(22) Date of filing: 06.03.2000
(51) International Patent Classification (IPC)7: A61K 31/437, A61K 31/435, A61K 31/495, A61K 31/497, A61K 31/498, A61K 31/506, A61K 31/517, A61K 31/541, A61K 31/5355, A61P 5/04, C07D 221/22, C07D 239/74, C07D 241/42, C07D 401/12, C07D 401/14, C07D 403/12, C07D 403/14, C07D 413/12
(86) International application number:
PCT/US0005/933
(87) International publication number:
WO 0053/181 (14.09.2000 Gazette 2000/37)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 10.03.1999 US 123640 P

(71) Applicant: Merck & Co., Inc.
Rahway, New Jersey 07065-0907 (US)

(72) Inventors:
  • WALSH, Thomas, F.
    Rahway, NJ 07065-0907 (US)
  • UJJAINWALLA, Feroze
    Rahway, NJ 07065-0907 (US)

(74) Representative: Horgan, James Michael Frederic 
Merck & Co., Inc., Terlings Park, Eastwick Road
Harlow, Essex CM20 2QR
Harlow, Essex CM20 2QR (GB)

   


(54) 6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE