DIBENZO-AZEPINE DERIVATIVES AS ALPHA V INTEGRIN RECEPTOR ANTAGONISTS - Patent 1169042

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EP 1 169 042 A1

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(43)	Date of publication:
	09.01.2002 Bulletin 2002/02

(21)	Application number: 00911811.8

(22)	Date of filing: 14.02.2000

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International Patent Classification (IPC)⁷: A61K 31/551, A61K 31/553, A61K 31/554, A61P 9/10, A61P 19/08, C07D 223/18, C07D 243/10, C07D 243/38, C07D 267/12, C07D 273/06, C07D 281/02, C07D 285/36, C07D 291/08, C07D 471/02, C07D 471/12, C07D 487/02, C07D 487/12, C07D 498/02, C07D 498/12, C07D 513/02, C07D 513/12

(86)	International application number:
	PCT/US0003/796

(87)	International publication number:
	WO 0048/603 (24.08.2000 Gazette 2000/34)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

17.02.1999 US 120564 P

(71)	Applicant: Merck & Co., Inc.
	Rahway, New Jersey 07065-0907 (US)

(72)	Inventors:
	PATANE, Michael, A. Rahway, NJ 07065-0907 (US) NEWTON, Randall, C. Rahway, NJ 07065-0907 (US)

(74)	Representative: Thompson, John Dr.
	Merck & Co., Inc. European Patent Department Terlings Park Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	DIBENZO-AZEPINE DERIVATIVES AS ALPHA V INTEGRIN RECEPTOR ANTAGONISTS