(19)

(11)

EP 1 185 511 A2

(12)

(88) Date of publication A3: 25.01.2001 (43) Date of publication: 13.03.2002 Bulletin 2002/11 (21) Application number: 00937698.9 (22) Date of filing: 24.05.2000

(51) International Patent Classification (IPC)7: C07D 207/16, C07D 211/60, C07C 311/39, C07D 403/04, C07D 401/04, C07D 413/04, C07D 243/08, C07D 241/04, A61P 7/00, A61K 31/40 (86) International application number: PCT/US0014/193 (87) International publication number: WO 0071/515 (30.11.2000 Gazette 2000/48)

(84) Designated Contracting States: AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE Designated Extension States: AL LT LV MK RO SI (30) Priority: 24.05.1999 US 135838 P (71) Applicant: COR THERAPEUTICS, INC. South San Francisco, CA 94080 (US)	(72) Inventors: ZHU, Bing-Yan Belmont, CA 94002 (US) SCARBOROUGH, Robert, M. Half Moon Bay, CA 94019 (US) (74) Representative: Clisci, Serge et al S.A. FEDIT-LORIOT & AUTRESCONSEILS EN PROPRIETE INDUSTRIELLE38, Avenue Hoche 75008 Paris 75008 Paris (FR)