IMIDAZO- AND PYRROLO[1,2-A]PYRIMID-4-ONES AS GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS - Patent 1185530

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EP 1 185 530 A1

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(43)	Date of publication:
	13.03.2002 Bulletin 2002/11

(21)	Application number: 00930676.2

(22)	Date of filing: 12.05.2000

(51)	International Patent Classification (IPC)⁷: C07D 487/04, A61K 31/505, A61P 15/00 // (C07D487/04, 209:00), C07D239:00,(C07D487/04, 235:00), C07D239:00

(86)	International application number:
	PCT/US0013/108

(87)	International publication number:
	WO 0069/859 (23.11.2000 Gazette 2000/47)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

14.05.1999 US 310878
28.07.1999 US 363254
23.09.1999 US 405286

(71)	Applicant: Neurocrine Biosciences, Inc.
	San Diego, CA 92121-1102 (US)

(72)	Inventors:
	ZHU, Yun-Fei San Diego, CA 92126 (US) WILCOXEN, Keith, M. San Diego, CA 92104 (US) STRUTHERS, R., Scott Encinitas, CA 92024 (US) CHEN, Chen San Diego, CA 92129 (US) CONNORS, Patrick, Jr. San Diego, CA 92014 (US) GAO, Yinghong San Diego, CA 92122 (US) TUCCI, Fabio, C. San Diego, CA 92121 (US)

(74)	Representative: Gowshall, Jonathan Vallance et al
	FORRESTER & BOEHMERTPettenkoferstrasse 20-22 80336 München 80336 München (DE)

(54)	IMIDAZO- AND PYRROLO[1,2-A]PYRIMID-4-ONES AS GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS