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<ep-patent-document id="EP1185535A1" country="EP" dtd-version="ep-patent-document-v1-4.dtd" doc-number="1185535" date-publ="20020313" file="00928691.5" lang="en" kind="A1" status="n"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYAL</B001EP><B003EP>*</B003EP><B005EP>X</B005EP><B007EP>DIM350 (Ver 2.1 Jan 2001) 1100000/0 1710000/0</B007EP></eptags></B000><B100><B110>1185535</B110><B130>A1</B130><B140><date>20020313</date></B140><B190>EP</B190></B100><B200><B210>00928691.5</B210><B220><date>20000501</date></B220><B240><B241><date>20011123</date></B241></B240><B250>En</B250><B251EP>En</B251EP><B260>En</B260></B200><B300><B310>183015 P</B310><B320><date>19990504</date></B320><B330><ctry>US</ctry></B330><B310>552036</B310><B320><date>20000419</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20020313</date><bnum>200211</bnum></B405><B430><date>20020313</date><bnum>200211</bnum></B430></B400><B500><B510><B516>7</B516><B511> 7C 07D 498/04   A</B511><B512> 7A 61K  31/535  B</B512><B512> 7A 61P  15/18   B</B512><B512> 7A 61P  35/00   B</B512><B514> 7C 07D 498/04   J</B514><B514> 7C 07D 333:00   J</B514><B515> 7C 07D 265:00   Z</B515><B517EP> // (C07D498/04, 333:00), C07D265:00</B517EP></B510><B540><B541>de</B541><B542>CYCLOCARBAMATE AND ZYCLISCHE AMIDODERIVATE</B542><B541>en</B541><B542>CYCLOCARBAMATE AND CYCLIC AMIDE DERIVATIVES</B542><B541>fr</B541><B542>CYCLOCARBAMATE ET DERIVES D'AMIDES CYCLIQUES</B542></B540></B500><B700><B710><B711><snm>American Home Products Corporation</snm><iid>00201465</iid><irf>00928691.5</irf><adr><str>Five Giralda Farms</str><city>Madison, New Jersey 07840</city><ctry>US</ctry></adr></B711><B711><snm>LIGAND PHARMACEUTICALS INCORPORATED</snm><iid>01034673</iid><irf>00928691.5</irf><adr><str>10275 Science Center Drive</str><city>San Diego,California 92121</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>SANTILLI, Arthur, A.</snm><adr><str>1737 Sue Ellen Drive</str><city>Havertown, PA 19083</city><ctry>US</ctry></adr></B721><B721><snm>VIET, Andrew, Q.</snm><adr><str>Apt. L-200,250 Beverly Boulevard</str><city>Upper Darby, PA 19082</city><ctry>US</ctry></adr></B721><B721><snm>ZHANG, Puwen</snm><adr><str>7004 Oriole Court</str><city>Audubon, PA 19403</city><ctry>US</ctry></adr></B721><B721><snm>FENSOME, Andrew</snm><adr><str>779 Trephanny Lane</str><city>Wayne, PA 19087</city><ctry>US</ctry></adr></B721><B721><snm>ZHI, Lin</snm><adr><str>7794 Roan Road</str><city>San Diego, CA 92129</city><ctry>US</ctry></adr></B721><B721><snm>JONES, Todd, K.</snm><adr><str>546 Marview Drive</str><city>Solana Beach, CA 92075</city><ctry>US</ctry></adr></B721><B721><snm>TEGLEY, Christopher, M.</snm><adr><str>478 Thunderhead Street</str><city>Thousand Oaks, CA 91360</city><ctry>US</ctry></adr></B721><B721><snm>WROBEL, Jay, E.</snm><adr><str>15 Rosetree Lane</str><city>Lawrenceville, NJ 08648</city><ctry>US</ctry></adr></B721><B721><snm>EDWARDS, James, P.</snm><adr><str>8723 Hesby Court</str><city>San Diego, CA 92129</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Hale, Stephen Geoffrey</snm><iid>00031411</iid><adr><str>JY &amp; GW Johnson,Kingsbourne House,229-231 High Holborn</str><city>London WC1V 7DP</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry></B840><B844EP><B845EP><ctry>AL</ctry><date>20011123</date></B845EP><B845EP><ctry>LT</ctry><date>20011123</date></B845EP><B845EP><ctry>LV</ctry><date>20011123</date></B845EP><B845EP><ctry>MK</ctry></B845EP><B845EP><ctry>RO</ctry><date>20011123</date></B845EP><B845EP><ctry>SI</ctry><date>20011123</date></B845EP></B844EP><B860><B861><dnum><anum>US0011825</anum></dnum><date>20000501</date></B861><B862>En</B862></B860><B870><B871><dnum><pnum>WO0066591</pnum></dnum><date>20001109</date><bnum>200045</bnum></B871></B870></B800></SDOBI></ep-patent-document>
