PREPARATION OF 7-SUBSTITUTED BENZOTHIOPHENES - Patent 1196413

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EP 1 196 413 A2

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(88)	Date of publication A3:
	19.07.2001

(43)	Date of publication:
	17.04.2002 Bulletin 2002/16

(21)	Application number: 00944592.5

(22)	Date of filing: 21.06.2000

(51)	International Patent Classification (IPC)⁷: C07D 409/04

(86)	International application number:
	PCT/US0011/884

(87)	International publication number:
	WO 0100/620 (04.01.2001 Gazette 2001/01)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

29.06.1999 US 141481 P

(71)	Applicant: ELI LILLY AND COMPANY
	Indianapolis, Indiana 46285 (US)

(72)	Inventors:
	MOHER, Eric, David Indianapolis, IN 46237 (US) O'TOOLE, John, Cunningham Indianapolis, IN 46221 (US) RIZZO, John, Robert Indianapolis, IN 46214 (US) VICENZI, Jeffrey, Thomas Brownsburg, IN 46112 (US) ZHANG, Tony, Yantao Indianapolis, IN 46236 (US)

(74)	Representative: Vaughan, Jennifer Ann et al
	Eli Lilly and Company LimitedLilly Research CentreErl Wood Manor Windlesham, Surrey GU20 6PH Windlesham, Surrey GU20 6PH (GB)

(54)	PREPARATION OF 7-SUBSTITUTED BENZOTHIOPHENES