1,2,3,4,5,6-HEXAHYDROAZEPINO 4,5-b]INDOLES CONTAINING ARYLSULFONES AT THE 9-POSITION

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EP 1 196 417 B8

(12)	CORRECTED EUROPEAN PATENT SPECIFICATION
	Note: Bibliography reflects the latest situation

(15)	Correction information:
	Corrected version no 1 (W1 B1)

(48)	Corrigendum issued on:
	15.06.2005 Bulletin 2005/24

(45)	Mention of the grant of the patent:
	20.04.2005 Bulletin 2005/16

(21)	Application number: 00946798.6

(22)	Date of filing: 11.07.2000

(51)	International Patent Classification (IPC)⁷: C07D 487/04, A61K 31/55, C07C 321/30, C07C 317/32, C07D 223/12 // (C07D487/04, 223:00), C07D209:00

(86)	International application number:
	PCT/US2000/016322

(87)	International publication number:
	WO 2001/005793 (25.01.2001 Gazette 2001/04)

(54)	1,2,3,4,5,6-HEXAHYDROAZEPINO 4,5-b]INDOLES CONTAINING ARYLSULFONES AT THE 9-POSITION 1,2,3,4,5,6,-HEXAHYDROAZEPINO[4,5-B]INDOLE, DIE ARYLSULFONE AN DIE 9-STELLUNG ENTHALTEN 1,2,3,4,5,6-HEXAHYDROAZEPINE 4,5-b]INDOLES CONTENANT DES ARYLSULFONES A LA POSITION 9

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

(30)

Priority:

19.07.1999 US 144574 P

(43)	Date of publication of application:
	17.04.2002 Bulletin 2002/16

(73)	Proprietor: Pharmacia & Upjohn Company LLC
	Kalamazoo, MI 49001 (US)

(72)	Inventors:
	JACOBSEN, E., Jon Kalamazoo, MI 49008 (US) HENDGES, Susan, K. Kalamazoo, MI 49006 (US)

(74)	Representative: Perry, Robert Edward
	GILL JENNINGS & EVERY Broadgate House 7 Eldon Street London EC2M 7LH London EC2M 7LH (GB)

(56)

References cited: :

EP-A- 0 013 414
EP-A- 0 028 381
EP-A- 0 102 476
EP-A- 0 354 303
EP-A- 0 666 253
WO-A-94/18980
WO-A-99/32463
WO-A-99/62506
DE-A- 2 120 708
DE-A- 2 438 120
DE-A- 2 548 910
DE-A- 2 748 978
DE-A- 3 831 445
DE-A- 19 829 357
FR-A- 1 499 717
FR-A- 2 110 283
FR-A- 2 154 568
FR-M- 6 699
JP-A- 2 048 564
US-A- 3 576 872
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US-A- 5 952 349

EP-A- 0 017 883
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CH-A- 619 460
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FR-A- 1 489 916
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GB-A- 1 293 540
JP-A- 60 044 557
US-A- 3 652 588
US-A- 3 948 987
US-A- 4 239 888
US-A- 4 332 820
US-A- 5 534 518

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