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<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIE......FI....CY..TR................................................</B001EP><B005EP>J</B005EP><B007EP>DIM360 Ver 2.15 (14 Jul 2008) -  2999001/0</B007EP></eptags></B000><B100><B110>1203766</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20120411</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>01125494.3</B210><B220><date>20011106</date></B220><B240><B241><date>20050323</date></B241><B242><date>20081103</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>707068</B310><B320><date>20001106</date></B320><B330><ctry>US</ctry></B330><B310>973142</B310><B320><date>20011009</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20120411</date><bnum>201215</bnum></B405><B430><date>20020508</date><bnum>200219</bnum></B430><B450><date>20120229</date><bnum>201209</bnum></B450><B452EP><date>20111014</date></B452EP><B480><date>20120411</date><bnum>201215</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 213/75        20060101AFI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 215/22        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07D 221/04        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07D 221/16        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>C07D 401/04        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>C07D 401/12        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>C07D 403/12        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>C07D 405/12        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>C07D 409/06        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 409/12        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="11"><text>C07D 409/14        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="12"><text>C07D 413/06        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="13"><text>C07D 413/12        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="14"><text>C07D 417/06        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="15"><text>C07D 471/04        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="16"><text>A61K  31/505       20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="17"><text>A61K  31/44        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="18"><text>A61K  31/50        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="19"><text>A61K  31/4704      20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="20"><text>A61P  29/00        20060101ALI20110823BHEP        </text></classification-ipcr><classification-ipcr sequence="21"><text>A61P  35/00        20060101ALI20110823BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>Carbonsäurederivate, die die Bindung von Integrinen an ihre Rezeptoren hemmen</B542><B541>en</B541><B542>Carboxylic acid derivatives that inhibit the binding of integrins to their receptors</B542><B541>fr</B541><B542>Dérivés d'acides carboxyliques inhibant la liaison des intégrines à leurs récepteurs</B542></B540><B560><B561><text>EP-A- 0 355 819</text></B561><B561><text>EP-A- 0 512 831</text></B561><B561><text>WO-A-00/67746</text></B561><B561><text>WO-A-00/68188</text></B561><B561><text>WO-A-01/46190</text></B561><B561><text>WO-A-91/13862</text></B561><B561><text>WO-A-96/22966</text></B561><B561><text>WO-A-99/52493</text></B561><B561><text>DE-A- 2 614 189</text></B561><B561><text>US-A- 5 484 946</text></B561><B561><text>US-A- 5 721 366</text></B561><B562><text>L. ISMAILI ET AL: "Synthesis of New Pyrazolo(4,3-c)quinoline-3-one Derivatives and some Oxazolo(4,5-c)quinoline-2,4-diones" JOURNAL OF HETEROCYCLIC CHEMISTRY, vol. 36, no. 3, 1999, pages 719-722, XP002298894</text></B562><B562><text>J.J. PANOUSE ET AL: "Relations structures-activités des immunomodulateurs. Apport de la modélisation moléculaire" ANNALES PHARMACEUTIQUES FRANCAISES, vol. 58, no. 5, 2000, pages 291-302, XP008036024</text></B562></B560></B500><B700><B720><B721><snm>Biediger, Ronald J.</snm><adr><str>17002 East Copper Lakes Court</str><city>Houston, TX  77095</city><ctry>US</ctry></adr></B721><B721><snm>Chen, Qi</snm><adr><str>2607 Parkbriar Lane</str><city>Pearland, TX 77584</city><ctry>US</ctry></adr></B721><B721><snm>Holland, George W.</snm><adr><str>402 Park Trail Lane</str><city>Houston, Texas 77007</city><ctry>US</ctry></adr></B721><B721><snm>Kassir, Jamal M.</snm><adr><str>310 Anne's Way,</str><city>Stafford, Texas 77477</city><ctry>US</ctry></adr></B721><B721><snm>Li, Wen</snm><adr><str>1954 Winrock,
Apt. 234</str><city>Houston, TX 77057</city><ctry>US</ctry></adr></B721><B721><snm>Market, Robert V.</snm><adr><str>2215 St. Jmaes Place</str><city>Pearland, TX 77581</city><ctry>US</ctry></adr></B721><B721><snm>Scott, Ian L.</snm><adr><str>25 Lea Drive</str><city>Delanson, NY 12053</city><ctry>US</ctry></adr></B721><B721><snm>Wu, Chengde</snm><adr><str>2511 Lansing Circle</str><city>Pearland, TX 77584</city><ctry>US</ctry></adr></B721><B721><snm>Decker, Radford E.</snm><adr><str>1078 West 42nd Street</str><city>Houston, TX 77018</city><ctry>US</ctry></adr></B721><B721><snm>Li, Jian</snm><adr><str>22 Wildflower Trace Place,
The Woodlands</str><city>Houston, TX 77382</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>ENCYSIVE PHARMACEUTICALS, INC.</snm><iid>101114597</iid><irf>J101183EP</irf><adr><str>235 East 42nd Street</str><city>New York, NY 10017</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Weber, Martin</snm><sfx>et al</sfx><iid>101202900</iid><adr><str>Jones Day 
Prinzregentenstraße 11</str><city>80538 München</city><ctry>DE</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry><ctry>TR</ctry></B840><B880><date>20041208</date><bnum>200450</bnum></B880></B800></SDOBI>
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