(19)
(11) EP 1 212 096 A2

(12)

(88) Date of publication A3:
31.01.2002

(43) Date of publication:
12.06.2002 Bulletin 2002/24

(21) Application number: 00959512.5

(22) Date of filing: 28.08.2000
(51) International Patent Classification (IPC)7A61K 47/48
(86) International application number:
PCT/US0023/593
(87) International publication number:
WO 0113/958 (01.03.2001 Gazette 2001/09)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 26.08.1999 US 150765 P
26.08.1999 US 150894 P
23.02.2000 US 184411 P
23.02.2000 US 184412 P

(71) Applicants:
  • Brenner, Sydney
    Berkeley, CA 94704 (US)
  • Goelet, Philip
    Baltimore, MD 21202 (US)
  • Stackhouse, Joseph
    Baltimore, MD 21202 (US)
  • Millward, Steven M.
    Baltimore, MD 21218 (US)

(72) Inventors:
  • Brenner, Sydney
    Berkeley, CA 94704 (US)
  • Goelet, Philip
    Baltimore, MD 21202 (US)
  • Stackhouse, Joseph
    Baltimore, MD 21202 (US)
  • Millward, Steven M.
    Baltimore, MD 21218 (US)

(74) Representative: Jump, Timothy John Simon et al
Venner Shipley & Co.20 Little Britain
London EC1A 7DH
London EC1A 7DH (GB)

   


(54) DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME