(19)
(11) EP 1 212 120 A2

(12)

(88) Date of publication A3:
28.02.2002

(43) Date of publication:
12.06.2002 Bulletin 2002/24

(21) Application number: 00962764.7

(22) Date of filing: 07.09.2000
(51) International Patent Classification (IPC)7A61P 35/00, A61K 31/135, A61K 31/235, A61K 31/33, A61K 31/519, A61K 31/4045, A61K 47/48
(86) International application number:
PCT/IB0001/427
(87) International publication number:
WO 0117/614 (15.03.2001 Gazette 2001/11)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 07.09.1999 US 152681 P

(71) Applicant: Conjuchem, Inc.
Montréal,Québec H2X 3Y8 (CA)

(72) Inventors:
  • BRIDON, Dominique, P.
    Ville Mont-Royal, Quebec H3P 2S2 (CA)
  • LEGER, Roger
    St-Lambert, Quebec J4R 2V8 (CA)
  • HUANG, Xicai
    Kirkland, Quebec H9J 3X2 (CA)
  • MILNER, Peter, G.
    Los Altos Hills, CA 94022 (US)
  • SMITH, Damon
    Westmount, Quebec H3Z 2E9 (CA)
  • EZRIN, Alan, M.
    Moraga, CA 94556 (US)

(74) Representative: Holmberg, Martin 
Bergenstrahle & Lindvall ABP.O. Box 17704
118 93 Stockholm
118 93 Stockholm (SE)

   


(54) METHODS AND COMPOSITIONS CONTAINING SUCCINIMIDE OR MALEIMIDE DERIVATIVES OF ANTINEOPLASTIC AGENTS, FOR PRODUCING LONG LASTING ANTINEOPLASTIC AGENTS