ARYLALKYLOXYALKYLAMINES AND ARYLALKYLTHIOALKYLAMINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NICOTINIC CHOLINERGIC RECEPTORS - Patent 1212301

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(11)

EP 1 212 301 A1

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(43)	Date of publication:
	12.06.2002 Bulletin 2002/24

(21)	Application number: 00945006.5

(22)	Date of filing: 30.06.2000

(51)	International Patent Classification (IPC)⁷: C07D 213/30, A61P 25/00, A61K 31/4406, C07D 213/61, C07D 213/65, C07D 215/20, C07D 239/26, C07D 453/02, C07D 213/32

(86)	International application number:
	PCT/US0017/978

(87)	International publication number:
	WO 0116/107 (08.03.2001 Gazette 2001/10)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

31.08.1999 US 387149

(71)	Applicant: Targacept, Inc.
	Winston-Salem, NC 27102-1487 (US)

(72)	Inventors:
	DULL, Gary Maurice Lewisville, NC 27023 (US) WAGNER, Jared Miller Durham, NC 27704 (US)

(74)	Representative: Bassett, Richard Simon
	Eric Potter Clarkson,Park View House,58 The Ropewalk Nottingham NG1 5DD Nottingham NG1 5DD (GB)

(54)	ARYLALKYLOXYALKYLAMINES AND ARYLALKYLTHIOALKYLAMINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NICOTINIC CHOLINERGIC RECEPTORS