HYDROXYALKANOYLAMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF ABETA PROTEIN PRODUCTION - Patent 1212306

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(11)

EP 1 212 306 A2

(12)

(88)	Date of publication A3:
	11.04.2002

(43)	Date of publication:
	12.06.2002 Bulletin 2002/24

(21)	Application number: 00963374.4

(22)	Date of filing: 13.09.2000

(51)	International Patent Classification (IPC)⁷: C07D 243/24, A61K 31/55, A61P 43/00, C07D 223/12, C07D 401/04, C07D 409/12, C07D 405/12, C07D 403/12, C07D 401/06

(86)	International application number:
	PCT/US0024/967

(87)	International publication number:
	WO 0119/797 (22.03.2001 Gazette 2001/12)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	LT LV RO SI

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Priority:

13.09.1999 US 153511 P
09.08.2000 US 224388 P

(71)	Applicant: BRISTOL-MYERS SQUIBB COMPANY
	Princeton, NJ 08543-4000 (US)

(72)	Inventors:
	OLSON, Richard, Eric Wilmington, DE 19803 (US) LIU, Hong Glen Mills, PA 18342 (US) THOMPSON, Lorin, Andrew, III Wilmington, DE 19809 (US)

(74)	Representative: Howard, Paul Nicholas et al
	Carpmaels & Ransford43 Bloomsbury Square London WC1A 2RA London WC1A 2RA (GB)

(54)	HYDROXYALKANOYLAMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF ABETA PROTEIN PRODUCTION