(19)
(11) EP 1 216 233 A1

(12)

(43) Date of publication:
26.06.2002 Bulletin 2002/26

(21) Application number: 00962482.6

(22) Date of filing: 13.09.2000
(51) International Patent Classification (IPC)7C07D 239/91, C07D 405/04, C07D 409/04, A61K 31/517, A61P 9/10
(86) International application number:
PCT/EP0008/939
(87) International publication number:
WO 0123/364 (05.04.2001 Gazette 2001/14)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 28.09.1999 US 407939

(71) Applicant: MERCK PATENT GmbH
64293 Darmstadt (DE)

(72) Inventors:
  • MEDERSKI, Werner
    64390 Erzhausen (DE)
  • DEVANT, Ralf
    64291 Darmstadt (DE)
  • BARNICKEL, Gerhard
    64298 Darmstadt (DE)
  • BERNOTAT-DANIELOWSKI, Sabine
    61231 Bad Nauheim (DE)
  • MELZER, Guido
    65719 Hofheim/Ts. (DE)
  • DHANOA, Daljit
    West Chester, PA 19382 (US)
  • ZHAO, Bao-Ping
    Plainsboro, NJ 08536 (US)
  • RINKER, James
    Kenhurst, PA 19607 (US)
  • PLAYER, Mark
    Phoenixville, PA 1946 (US)
  • SOLL, Richard
    Lawrenceville, NJ 08648 (US)
  • CEZANNE, Bertram
    D-64546 Mörfelden-Walldorf (DE)

   


(54) QUINAZOLINONES