PYRAZOLOANTHRONE AND DERIVATIVES THEREOF AS JNK INHIBITORS AND THEIR COMPOSITIONS - Patent 1218347

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EP 1 218 347 A1

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(43)	Date of publication:
	03.07.2002 Bulletin 2002/27

(21)	Application number: 00955709.1

(22)	Date of filing: 19.08.2000

(51)	International Patent Classification (IPC)⁷: C07D 231/54, C07D 401/04, C07D 413/04, C07D 401/12, C07D 409/12, A61K 31/415

(86)	International application number:
	PCT/US0022/727

(87)	International publication number:
	WO 0112/609 (22.02.2001 Gazette 2001/08)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

19.08.1999 US 378234

(71)	Applicant: SIGNAL PHARMACEUTICALS, INC.
	San Diego, CA 92121 (US)

(72)	Inventors:
	BENNETT, Brydon, L. San Diego, CA 92117 (US) BHAGWAT, Shripad, S. San Diego, CA 92130 (US) MANNING, Anthony, M. San Diego, CA 92129 (US) MURRAY, Brion, W. San Diego, CA 92106 (US) O'LEARY, Eoin, C. San Diego, CA 92116 (US) SATOH, Yoshitaka San Diego, CA 92131 (US)

(74)	Representative: Jump, Timothy John Simon et al
	Venner Shipley & Co.20 Little Britain London EC1A 7DH London EC1A 7DH (GB)

(54)	PYRAZOLOANTHRONE AND DERIVATIVES THEREOF AS JNK INHIBITORS AND THEIR COMPOSITIONS