TETRAHYDROBENZINDOLONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS 5-HT7 RECEPTOR ANTAGONISTS - Patent 1222185

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EP 1 222 185 A1

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(43)	Date of publication:
	17.07.2002 Bulletin 2002/29

(21)	Application number: 00971384.3

(22)	Date of filing: 13.10.2000

(51)	International Patent Classification (IPC)⁷: C07D 403/12, C07D 413/12, C07D 417/12, C07D 401/14, A61K 31/445, A61K 31/495, A61K 31/44, A61P 25/00

(86)	International application number:
	PCT/EP0010/149

(87)	International publication number:
	WO 0129/029 (26.04.2001 Gazette 2001/17)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

18.10.1999 GB 9924628
14.03.2000 GB 0006168
03.08.2000 GB 0018952

(71)	Applicant: SMITHKLINE BEECHAM PLC
	Brentford,Middlesex TW8 9EP (GB)

(72)	Inventors:
	BROMIDGE, Steven MarkSmithKline Beecham Pharmac. HarlowEssex CM19 5AW (GB) GRIBBLE, Andrew D.SmithKline Beecham Pharmaceu. HarlowEssex CM19 5AW (GB) LOVELL, Peter JohnSmithKline Beecham Pharmaceu. HarlowEssex CM19 5AW (GB) WITHERINGTON, JasonSmithkline Beecham Pharmac. HarlowEssex CM19 5AW (GB)

(74)	Representative: Giddings, Peter John, Dr.
	GlaxoSmithKlineCorporate Intellectual Property (CN9.25.1)980 Great West Road Brentford, Middlesex TW8 9GS Brentford, Middlesex TW8 9GS (GB)

(54)	TETRAHYDROBENZINDOLONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS 5-HT7 RECEPTOR ANTAGONISTS