(19)
(11) EP 1 226 112 A2

(12)

(88) Date of publication A3:
13.09.2001

(43) Date of publication:
31.07.2002 Bulletin 2002/31

(21) Application number: 00982697.5

(22) Date of filing: 18.10.2000
(51) International Patent Classification (IPC)7C07C 233/00, A01N 37/18
(86) International application number:
PCT/US0041/248
(87) International publication number:
WO 0128/498 (26.04.2001 Gazette 2001/17)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 18.10.1999 US 160033 P

(71) Applicant: THE UNIVERSITY OF CONNECTICUT
Farmington, CT 06030 (US)

(72) Inventors:
  • MAKRIYANNIS, Alexandros
    Willimantic, CT 06226 (US)
  • LIU, Qian
    Storrs, CT (US)
  • GOUTOPOULOS, Andreas
    Boston, MA 02116 (US)

(74) Representative: Beacham, Annabel Rose et al
Frank B. Dehn & Co.,European Patent Attorneys,179 Queen Victoria Street
London EC4V 4EL
London EC4V 4EL (GB)

   


(54) RETRO-ANANDAMIDES, HIGH AFFINITY AND STABILITY CANNABINOID RECEPTOR LIGANDS