BETA-AMINOACID COMPOUNDS USEFUL FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS - Patent 1230220

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EP 1 230 220 A1

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(43)	Date of publication:
	14.08.2002 Bulletin 2002/33

(21)	Application number: 00978213.7

(22)	Date of filing: 26.10.2000

(51)	International Patent Classification (IPC)⁷: C07D 223/18, C07D 223/16, C07D 243/12, C07D 243/24, C07D 267/14, C07D 281/10, C07D 487/04, A61K 31/5513, A61K 31/5517, A61K 31/551, A61K 31/554, A61P 25/28 // (C07D487/04, 243:00), C07D209:00

(86)	International application number:
	PCT/US0026/278

(87)	International publication number:
	WO 0134/571 (17.05.2001 Gazette 2001/20)

(84)	Designated Contracting States:
	AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV MK RO SI

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Priority:

09.11.1999 US 164399 P

(71)	Applicant: ELI LILLY AND COMPANY
	Indianapolis, Indiana 46285 (US)

(72)	Inventors:
	AUDIA, James, Edmund Indianapolis, IN 46278 (US) PORTER, Warren, Jaye Indianapolis, IN 46260 (US) SCOTT, William, Leonard Indianapolis, IN 46208 (US) STACK, Douglas, Richard Fishers, IN 46038 (US) THOMPSON, Richard, Craig Frankfort, IN 46041 (US)

(74)	Representative: Pritchard, Judith et al
	Eli Lilly and Company LimitedLilly Research CentreErl Wood ManorSunninghill Road Windlesham, Surrey GU20 6PH Windlesham, Surrey GU20 6PH (GB)

(54)	BETA-AMINOACID COMPOUNDS USEFUL FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS