(19)

(11)

EP 1 231 957 A1

(12)

(43) Date of publication: 21.08.2002 Bulletin 2002/34 (21) Application number: 00963532.7 (22) Date of filing: 14.09.2000

(51) International Patent Classification (IPC)7: A61M 5/00, B67D 5/08 (86) International application number: PCT/US0025/411 (87) International publication number: WO 0101/9432 (22.03.2001 Gazette 2001/12)

(84) Designated Contracting States: AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE Designated Extension States: AL LT LV MK RO SI (30) Priority: 14.09.1999 US 395363 31.01.2000 US 494387 (71) Applicant: Pharmacopeia Inc. Princeton, NJ 08543-5350 (US)	(72) Inventor: FEYGIN, Ilya Mountainside, NJ 07092 (US) (74) Representative: Musker, David Charles et al R.G.C. Jenkins & Co.26 Caxton Street London SW1H 0RJ London SW1H 0RJ (GB)