(19)
(11) EP 1 235 795 A1

(12)

(43) Date of publication:
04.09.2002 Bulletin 2002/36

(21) Application number: 00976591.8

(22) Date of filing: 03.11.2000
(51) International Patent Classification (IPC)7C07C 303/34, C07D 263/26, C07C 307/10
(86) International application number:
PCT/US0028/877
(87) International publication number:
WO 0103/6383 (25.05.2001 Gazette 2001/21)
(84) Designated Contracting States:
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 18.11.1999 GB 9927302

(71) Applicant: ELI LILLY AND COMPANY
Indianapolis, Indiana 46285 (US)

(72) Inventors:
  • ANTOINE, Luc, Jean, Jules
    B-3401 Landen (BE)
  • BORGHESE, Alfio
    B-1470 Baisy-Thy (BE)
  • VAN HOECK, Jean-Pierre, Joseph, Sylvain
    B-1475 Chastre (BE)

(74) Representative: Vaughan, Jennifer Ann 
Eli Lilly and Company LimitedLilly Research CentreErl Wood Manor
Windlesham, Surrey GU20 6PH
Windlesham, Surrey GU20 6PH (GB)

   


(54) PROCESS FOR THE PREPARATION OF SULFAMIDES